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熊去氧胆酸(ursodeoxycholic Acid)国际专利 

 

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ursodeoxycholic Acid 熊去氧胆酸欧洲专利

1  PROCESS FOR PREPARING URSODEOXYCHOLIC ACID DI-SODIUM 3,7-DISULFATE in my patents list  
   Inventor: FERRARI MASSIMO (IT); BONALDI MATTEO (IT); (+1)  Applicant: ERREGIERRE SPA (IT)
   EC:  C07J9/00; C07J31/00 IPC: C07J9/00; C07J31/00; C07J9/00 (+3)
   Publication info: EP1618121 - 2006-01-25
 
2  NITROSATED AND/OR NITROSYLATED URSODEOXYCHOLIC ACID COMPOUNDS, COMPOSITIONS AND METHODS OF USE in my patents list  
   Inventor: GARVEY DAVID S (US); IYENGAR RADHA (US)  Applicant: NITROMED INC (US); GARVEY DAVID S (US); (+1)
   EC:  C07J41/00C8 IPC: C07J41/00; C07J41/00; (IPC1-7): A61K 
   Publication info: WO2004012686 - 2004-02-12
 
3  A PROCESS FOR PREPARING URSODEOXYCHOLIC ACID DUSULPHATE AND PHARMACEUTICALLY ACCEPTABLE SALTS THEREOF in my patents list  
   Inventor: GIRAUDI ALBERTO (IT)  Applicant: ABC INTERNAT PHARMA S R L (IT); GIRAUDI ALBERTO (IT)
   EC:  C07J31/00C IPC: C07J31/00; C07J31/00; (IPC1-7): C07J31/00 
   Publication info: WO03066657 - 2003-08-14
 
4  Microgranules of Ursodeoxycholic acid in my patents list  
   Inventor: CECCHETELLI LOREDANA (IT); DI RELLA MARIO (IT); (+1)  Applicant: ISTITUTO BIOCHIMICO ITALIANO (IT)
   EC:  A61K9/00M18B; A61K9/00N2; (+3) IPC: A61K9/00; A61K9/16; A61K9/20 (+7)
   Publication info: EP1317925 - 2003-06-11
 
5  PROPHYLACTIC/THERAPEUTIC AGENT FOR LARGE INTESTINAL TUMOR, CONTAINING URSODEOXYCHOLIC ACID DERIVATIVE AS ACTIVE INGREDIENT in my patents list  
   Inventor: NARISAWA TOMIO  Applicant: MITSUBISHI PHARMA CORP
   EC:  IPC: A61K31/575; A61P35/00; C07J9/00 (+6)
   Publication info: JP2003012519 - 2003-01-15
 
6  USE OF URSODEOXYCHOLIC ACID FOR POTENTIATION OF THE PHOTOTOXIC EFFECT OF PHOTODYNAMIC THERAPY in my patents list  
   Inventor: KESSEL DAVID (US); REINERS JOHN J (US)  Applicant: UNIV WAYNE STATE (US); KESSEL DAVID (US); (+1)
   EC:  A61K31/575; A61K41/00W IPC: A61K31/575; A61K41/00; A61K31/575 (+2)
   Publication info: WO0182860 - 2001-11-08
 
7  A method for rendering ursodeoxycholic acid in soluble form pharmaceutical compositions in my patents list  
   Inventor: OLIVIERI ALDO (IT)  Applicant: BIOPROGRESS SPA (IT)
   EC:  A61K31/575; A61K47/48W18B; (+1) IPC: A61K31/575; A61K47/48; A61K31/575 (+4)
   Publication info: EP1147779 - 2001-10-24

8  TERTIARY AMINE SALT OF URSODEOXYCHOLIC ACID AND METHOD FOR PRODUCING URSODEOXYCHOLIC ACID USING THE SAME in my patents list  
   Inventor: MIKAMI KAZUTOSHI; KIMURA NORIYUKI; (+2)  Applicant: MITSUBISHI TOKYO PHARM INC
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP2001261696 - 2001-09-26
 
9  BUDESONIDE ALONE OR IN COMBINATION WITH URSODEOXYCHOLIC ACID IN THE THERAPY OF CHOLESTATIC LIVER DISEASES in my patents list  
   Inventor: LEUSCHNER MARIA  Applicant: FALK PHARMA GMBH (DE)
   EC:  A61K31/58 IPC: A61K31/58; A61K31/58; (IPC1-7): A61K31/00 
   Publication info: WO9916429 - 1999-04-08
 
10  URSODEOXYCHOLIC ACID DERIVATIVES AND METHODS FOR PRODUCING THEM in my patents list  
   Inventor: OKUMOTO HIROSHI (JP); NAKANISHI KATSUYOSHI (JP); (+5)  Applicant: KAKEN PHARMA CO LTD (JP); BIO RES CORP OF YOKOHAMA (JP); (+1)
   EC:  IPC: C07J9/00; C07J17/00; C07J75/00 (+5)
   Publication info: CA2237076 - 1999-07-08
 
11  PURIFICATION OF URSODEOXYCHOLIC ACID OR CHENODEOXYCHOLIC ACID in my patents list  
   Inventor: KAMIYAMA FUMIO; YAMAZAKI KAZUTOSHI; (+1)  Applicant: SEKISUI CHEMICAL CO LTD
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP56059796 - 1981-05-23

12  USE OF URSODEOXYCHOLIC ACID FOR THE TOPICAL TREATMENT OF INFLAMMATORY DISEASES OF THE MUCOUS MEMBRANES in my patents list  
   Inventor: TAUSCHEL HORST-DIETMAR (DE)  Applicant: FALK PHARMA GMBH (DE); TAUSCHEL HORST DIETMAR (DE)
   EC:  A61K31/575 IPC: A61K31/575; A61K31/575; (IPC1-7): A61K31/575 
   Publication info: WO9818474 - 1998-05-07
 
13  USE OF URSODEOXYCHOLIC ACID IN HIV INFECTION in my patents list  
   Inventor: SCHENTKE KLAUS-ULRICH (DE); KUERKTSCHIEV DIMO (DE)  Applicant: FALK PHARMA GMBH (DE); SCHENTKE KLAUS ULRICH (DE); (+1)
   EC:  A61K31/575 IPC: A61K31/575; A61K31/575; (IPC1-7): A61K31/575 
   Publication info: WO9805339 - 1998-02-12
 
14  COMBINATIONS OF AN URSODEOXYCHOLIC ACID COMPOUND AND A NSAID FOR THE CHEMOPREVENTIVE PROTECTION OF THE COLORECTUM in my patents list  
   Inventor: LARSON MARK V; AHLQUIST DAVID A; (+1)  Applicant: MAYO FOUNDATION (US)
   EC:  A61K31/575; A61K31/60; (+1) IPC: A61K31/575; A61K31/60; A61K45/06 (+8)
   Publication info: WO9734608 - 1997-09-25
 
15  SULFATE CONJUGATES OF URSODEOXYCHOLIC ACID, AND THEIR BENEFICIAL USE IN INFLAMMATORY DISORDERS AND OTHER APPLICATIONS in my patents list  
   Inventor: SETCHELL KENNETH D R  Applicant: CHILDRENS HOSP MEDICAL CENTER (US)
   EC:  A61K31/575 IPC: A61K31/575; A61K31/575; (IPC1-7): A61K31/575 
   Publication info: WO9718816 - 1997-05-29

16  THERAPEUTIC AGENT FOR LACTOSE INTOLERANCE CONTAINING URSODEOXYCHOLIC ACID AS ACTIVE INGREDIENT in my patents list  
   Inventor: YAKIDA AKIKUNI  Applicant: YAKIDA AKIKUNI; TOKYO TANABE CO
   EC:  IPC: A61K31/575; C07J1/00; A61K31/575 (+3)
   Publication info: JP9124689 - 1997-05-13
 
17  URSODEOXYCHOLIC ACID DERIVATIVE in my patents list  
   Inventor: TAKAHASHI MAKOTO; OTA SHUNSAKU; (+1)  Applicant: KAKEN PHARMA CO LTD; TAKAHASHI MAKOTO; (+1)
   EC:  IPC: A61K31/16; C07J1/00; A61K31/16 (+3)
   Publication info: JP9095496 - 1997-04-08
 
18  MEDICINE COMPOSITION COMPOUNDED WITH URSODEOXYCHOLIC ACID in my patents list  
   Inventor: YAKIDA AKIKUNI  Applicant: YAKIDA AKIKUNI; TOKYO TANABE CO
   EC:  IPC: A61K31/575; A61K38/46; A61K31/575 (+3)
   Publication info: JP9020679 - 1997-01-21
 
19  LIQUID-DOSAGE TYPE MEDICINE CONTAINING URSODEOXYCHOLIC ACID in my patents list  
   Inventor: YOOZEFU ORAFU BUIDAUERU  Applicant: MEDICHEMIE AG
   EC:  A61K9/00N2; A61K31/575 IPC: A61K9/00; A61K31/575; A61K9/00 (+6)
   Publication info: JP7082150 - 1995-03-28
 
20  Pharmaceutical compositions containing ursodeoxycholic acid. in my patents list  
   Inventor: OLIVIERI ALDO (IT); CAMPONESCHI CLAUDIO (IT)  Applicant: BIOPROGRESS SPA (IT)
   EC:  A61K9/16H6B; A61K9/16H6F; (+1) IPC: A61K9/16; A61K31/575; A61K9/16 (+3)
   Publication info: EP0599282 - 1994-06-01
 
21  PRODUCTION OF URSODEOXYCHOLIC ACID in my patents list  
   Inventor: HATTORI MASAHIKO; MIKAMI KAZUTOSHI  Applicant: TOKYO TANABE CO
   EC:  IPC: A61K31/575; C07J9/00; C25B3/04 (+7)
   Publication info: JP6002184 - 1994-01-11
 
22  Chenodeoxycholic acid or ursodeoxycholic acid for the treatment of diseases of the respiratory organs. in my patents list  
   Inventor: WIDAUER JOSEF OLAF DR MED (CH)  Applicant: MEDICHEMIE AG (CH)
   EC:  A61K31/575 IPC: A61K31/575; A61K31/575; (IPC1-7): A61K31/575 
   Publication info: EP0514328 - 1992-11-19
 
23  LONG ACTING PREPARATION OF URSODEOXYCHOLIC ACID in my patents list  
   Inventor: TAGUMA KAZUNORI; YAZAKI TAKASHI; (+2)  Applicant: TOKYO TANABE CO
   EC:  IPC: A61K9/14; A61K31/575; C07J9/00 (+7)
   Publication info: JP6024991 - 1994-02-01
 
24  NOVEL URSODEOXYCHOLIC ACID DERIVATIVE in my patents list  
   Inventor: SCOLASTICO CARLO (IT); PALAZZI CAMILLO MARIA FRANCESC (IT)  Applicant: ISTITUTO CHEMIOTERAPICO (IT)
   EC:  C07J51/00 IPC: C07J51/00; C07J51/00; (IPC1-7): C07J51/00 (+1)
   Publication info: WO9000175 - 1990-01-11
 
25  Phosphoric di-ester of ursodeoxycholic acid and its derivatives, process for their preparation and therapeutic compositions which contain them as active substances in my patents list  
   Inventor: PURICELLI LAURA  Applicant: MAGIS FARMACEUTICI (IT)
   EC:  IPC: A61K; (IPC1-7): A61K 
   Publication info: IT1226144 - 1990-12-19
 
26  Process for the preparation of the magnesium double salt of chenodeoxycholic acid and ursodeoxycholic acid in my patents list  
   Inventor: AIGNER ARNO DIPL CHEM DR (DE); BAUER ADOLF DIPL CHEM DR (DE); (+2)  Applicant: DIAMALT AG (DE)
   EC:  C07J51/00 IPC: C07J51/00; C07J51/00; (IPC1-7): C07J9/00 
   Publication info: DE3742798 - 1989-06-29
 
27  Process for preparing ursodeoxycholic acid derivates and their inorganic and organic salts having therpeutic activity. in my patents list  
   Inventor: REINER ALBERTO  Applicant: JAGO RES AG (CH)
   EC:  C07J41/00C8A IPC: C07J41/00; C07J41/00; (IPC1-7): A61K31/575 (+1)
   Publication info: EP0272462 - 1988-06-29
 
28  Process for preparing therapeutically active derivatives of ursodeoxycholic acid. in my patents list  
   Inventor: REINER ALBERTO  Applicant: JAGO RES AG (CH)
   EC:  C07J31/00C; C07J41/00C8 IPC: C07J31/00; C07J41/00; C07J31/00 (+4)
   Publication info: EP0273188 - 1988-07-06
 
29  Pharmaceutical compositions containing ursodeoxycholic acid. in my patents list  
   Inventor: POUPON RAOUL  Applicant: SYNTHELABO (FR)
   EC:  A61K31/575 IPC: A61K31/575; A61K31/575; (IPC1-7): A61K31/575 
   Publication info: EP0269516 - 1988-06-01

30  PRODUCTION OF 5'-URSODEOXYCHOLIC ACID in my patents list  
   Inventor: KUBOTA NAOHIRO  Applicant: ADEKA ARGUS CHEMICAL CO LTD
   EC:  IPC: C07J9/00; C07J75/00; C07J9/00 (+2)
   Publication info: JP1061496 - 1989-03-08
 
31  PRODUCTION OF URSODEOXYCHOLIC ACID in my patents list  
   Inventor: NIHEI TAKUYA; HAGA TAKASHI  Applicant: TOYO TIRE & RUBBER CO
   EC:  IPC: C12P33/06; C12R1/77; C12P33/00 (+2)
   Publication info: JP62122595 - 1987-06-03
 
 
32  Ursodeoxycholic acid derivative, process for its preparation, and pharmaceutical composition containing such a derivative in my patents list  
   Inventor: MASSAROLI GIANGIACOMO DR (IT)  Applicant: POLI IND CHIMICA SPA (IT)
   EC:  C07D321/00; C07J9/00B IPC: C07D321/00; C07J9/00; C07D321/00 (+3)
   Publication info: DE3433188 - 1985-03-28
 
33  PREPARATION OF URSODEOXYCHOLIC ACID BY EDIBLE BASIDIOMYCETES in my patents list  
   Inventor: TERADA MASAKI; HORIE YOSHIAKI; (+4)  Applicant: NISSIN FOOD PRODUCTS LTD
   EC:  IPC: C12P33/02; C12R1/645; C12P33/00 (+2)
   Publication info: JP60172296 - 1985-09-05
 
34  URSODEOXYCHOLIC ACID MEGLUMINE SALT AND INJECTION CONTAINING SAME in my patents list  
   Inventor: SUZUKI TADAYUKI; YANAGIHARA HIROYUKI; (+1)  Applicant: TOKYO TANABE CO
   EC:  IPC: A61K9/08; A61K31/13; A61K31/575 (+9)
   Publication info: JP60163897 - 1985-08-26
 
35  CHENODEOXYCHOLIC ACID OR URSODEOXYCHOLIC ACID DERIVATIVE, PREPARATION THEREOF AND MEDICINE CONTAINING SAME in my patents list  
   Inventor: ITOU MASAHARU; YAMATSU ISAO; (+4)  Applicant: EISAI CO LTD
   EC:  IPC: A61K31/575; C07J9/00; A61K31/575 (+3)
   Publication info: JP60161996 - 1985-08-23
 
36  Magnesium salt of chenodeoxycholic acid and ursodeoxycholic acid, the process for its preparation, and therapeutic compositions which contain it as active principle. in my patents list  
   Inventor: GARZIA ALDO; BOTTAZZI ANDREA  Applicant: ISTITUTO CHEMIOTERAPICO (IT)
   EC:  C07J9/00B; C07J51/00 IPC: C07J9/00; C07J51/00; C07J9/00 (+4)
   Publication info: EP0092073 - 1983-10-26
 
37  A method for producing ursodeoxycholic acid. in my patents list  
   Inventor: SAWADA HARUJI; TAGUCHI HISAHARU  Applicant: YAKULT HONSHA KK (JP)
   EC:  C07J9/00B; C12P33/06 IPC: C07J9/00; C12P33/06; C07J9/00 (+3)
   Publication info: EP0088637 - 1983-09-14
 
38  Aqueous solution of ursodeoxycholic acid for therapeutic uses, process for its preparation and its utilization for the treatment of cholelithiasis. in my patents list  
   Inventor: LARUELLE CLAUDE; LEPANT MARCEL  Applicant: PANMEDICA SA (FR)
   EC:  A61K31/575; C07J9/00B IPC: A61K31/575; C07J9/00; A61K31/575 (+4)
   Publication info: EP0086705 - 1983-08-24

39  PRODUCTION OF URSODEOXYCHOLIC ACID in my patents list  
   Inventor: TAGUCHI ISAMU  Applicant: SHOWA DENKO KK
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP59139399 - 1984-08-10

40  PROCESS FOR PREPARING HIGH PURITY URSODEOXYCHOLIC ACID in my patents list  
   Inventor:   Applicant: ERREGIERRE SPA (IT)
   EC:  C07J9/00B; C07J51/00 IPC: C07J9/00; C07J51/00; C07J9/00 (+2)
   Publication info: PT74749 - 1982-05-01
 
41  PURE URSODEOXYCHOLIC ACID BY NOVEL SYNTHETIC ROUTE in my patents list  
   Inventor:   Applicant: ERREGIERRE SPA
   EC:  C07J9/00B; C07J51/00 IPC: C07J9/00; C07J51/00; C07J9/00 (+2)
   Publication info: GB2076823 - 1981-12-09
 
42  PRODUCTION OF CRUDE URSODEOXYCHOLIC ACID in my patents list  
   Inventor: TAKEDA HARUKI; YABE MASAHIRO  Applicant: TOKYO TANABE CO
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP57056499 - 1982-04-05
 
43  PRODUCTION OF CRUDE URSODEOXYCHOLIC ACID in my patents list  
   Inventor: TAKEDA HARUKI  Applicant: TOKYO TANABE CO
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP57056498 - 1982-04-05
 
44  PRODUCTION OF CRUDE URSODEOXYCHOLIC ACID in my patents list  
   Inventor: TAKEDA HARUKI  Applicant: TOKYO TANABE CO
   EC:  IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP57056497 - 1982-04-05
 
45  HIGHLY PURE URSODEOXYCHOLIC ACID AND A PROCESS FOR PRODUCING IT in my patents list  
   Inventor:   Applicant: ROUSSEL UCLAF
   EC:  C07J9/00B IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: GB2052507 - 1981-01-28

46  NOVEL MANUFACTURE OF URSODEOXYCHOLIC ACID in my patents list  
   Inventor: ARUMAN GIIYUMETSUTO; ABERU FURANSOWA  Applicant: ROUSSEL UCLAF
   EC:  C07J9/00B IPC: C07J9/00; C07J9/00; (IPC1-7): C07J9/00 
   Publication info: JP55085600 - 1980-06-27
 


ursodeoxycholic Acid 熊去氧胆酸美国专利

 PAT. NO.  Title
1 6,297,229  Use of ursodeoxycholic acid to treat nonalcoholic steatohepatitis
2 6,251,884  Sulfate conjugates of ursodeoxycholic acid, and their beneficial use in inflammatory disorders and other applications
3 6,075,132  Ursodeoxycholic acid derivatives and methods for producing them
4 5,858,998  Budesonide alone or in combination with ursodeoxycholic acid in the therapy of cholestatic liver diseases
5 5,763,435  Sulfate conjugates of ursodeoxycholic acid, and their beneficial use in inflammatory disorders
6 5,534,505  Ursodeoxycholic acid-containing medicament in a liquid adminstration form
7 4,865,765  Ursodeoxycholic acid derivatives and their inorganic and organic salts having therapeutic activity, and process for preparing the same
8 4,828,763  Therapeutically active derivatives of ursodeoxycholic acid and process for preparing the same
9 4,579,819  Method for production of ursodeoxycholic acid by means of microbial transformation
10 4,547,271  Process for the electrochemical reduction of 7-ketolithocholic acid to ursodeoxycholic acid
11 4,440,688  Novel derivatives of ursodeoxycholic acid
12 4,379,093  Process for preparing high purity ursodeoxycholic acid
13 4,337,206  Process for preparing high purity ursodeoxycholic acid
14 4,316,848  Process for the purification of ursodeoxycholic acid
15 4,185,099  Hair and scalp treatment with compositions containing chenodeoxycholic or ursodeoxycholic acid
16 20040029965 Formulations for reducing or eliminating toxicity of enviromental hormones containing ursodeoxycholic acid 

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